Difference between revisions of "Other ergolines"
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(it still unknown if these can cause gangreen / nercosis in certain people..) | (it still unknown if these can cause gangreen / nercosis in certain people..) | ||
| − | -(s)Lasba : a(stereoseective butyl analoog | + | -(s)Lasba : a(stereoseective butyl analoog on the 8-amide) has been found active in humans, but mostly act as a stimulant (perdue uni/nichols/personal exprience) |
nice info to be found here : [http://bitnest.ca/Silo42/10.1007/BF02245940.pdf] | nice info to be found here : [http://bitnest.ca/Silo42/10.1007/BF02245940.pdf] | ||
| − | -also the morpholine and methyl-ethyl-amide moity are active ( | + | -also the morpholine and methyl-ethyl-amide moity are active (hoffman/stoll at sandoz, and shulgin mentions it in Tihkal.) |
promising : | promising : | ||
- future research is being done to replace the carboxylic acid to a "thoiacid" (actually a thioeaster) | - future research is being done to replace the carboxylic acid to a "thoiacid" (actually a thioeaster) | ||
| − | this means | + | this means at the top the oxygen will be repaced with a sulphur(=thio) and then still have room for the N-diethyl amide. (activity of these compound are still unknown.) |
- non-psychoactive ergolines : | - non-psychoactive ergolines : | ||
Revision as of 12:42, 11 March 2014
Other ergolines
on the 8 position :
- some of the lysergic precursors : methysergide, ergometrine and metyl-ergmetrine are slightly active above 1 mg. source (J.ott in Pharmacotheon )
(it still unknown if these can cause gangreen / nercosis in certain people..)
-(s)Lasba : a(stereoseective butyl analoog on the 8-amide) has been found active in humans, but mostly act as a stimulant (perdue uni/nichols/personal exprience) nice info to be found here : [1]
-also the morpholine and methyl-ethyl-amide moity are active (hoffman/stoll at sandoz, and shulgin mentions it in Tihkal.)
promising : - future research is being done to replace the carboxylic acid to a "thoiacid" (actually a thioeaster)
this means at the top the oxygen will be repaced with a sulphur(=thio) and then still have room for the N-diethyl amide. (activity of these compound are still unknown.)
- non-psychoactive ergolines :
bromocryptine, dihydroergotamine , dihydrolysergic, carbagoline and a bunch more , now used as proper migrane- an other-medicine.
on the 6 position : AL-LAD, BU-LAD, CYP-LAD, ETH-LAD, PRO-LAD and a few others, Mostly developed by Nichols but in coalition with Shulgin.
